SCHEMBL140753

SCHEMBL140753

Cc1cc(C)c(CNS(=O)(=O)C(F)(F)F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.42
PTGS2 P35354 2/20 0.42
CA2 P00918 3/20 0.39
CA1 P00915 2/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
CA12 O43570 1/20 0.35
CA7 P43166 1/20 0.35
CA13 Q8N1Q1 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
GRIA4 P48058 1/20 0.34
HTT P42858 2/20 0.33
FFAR4 Q5NUL3 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL138442 0.92 PTGS1 (0.44) PTGS1PTGS2CA2CA1MMP1
SCHEMBL140649 0.78 PTGS1 (0.47) PTGS1PTGS2CA2CA1GRIA4
SCHEMBL13090062 0.77 CA2 (0.42) PTGS1PTGS2CA2CA1MAPT
SCHEMBL139599 0.73 PTGS1 (0.51) PTGS1PTGS2CA2CA1MAPT
SCHEMBL139635 0.72 PTGS1 (0.59) PTGS1PTGS2CA2CA1MAPT
SCHEMBL138380 0.71 CA2 (0.47) PTGS1PTGS2CA2CA1GRIA4
SCHEMBL139634 0.70 PTGS1 (0.46) PTGS1PTGS2CA2CA1MAPT
SCHEMBL20847614 0.68 RAPGEF4 (0.35) LMNARAPGEF4ALDH1A1
SCHEMBL141067 0.68 CA2 (0.65) CA2CA1CA12CYP1A2CYP3A4
SCHEMBL27529567 0.67 CA1 (0.37) CA2CA1MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059179-A1 PALLADIUM-CATALYZED ORTHO-FLUORINATION The Scripps Research Insitiute (US) 2012-03-08 US disclosed
WO-2010115098-A2 PALLADIUM-CATALYZED ORTHO-FLUORINATION THE SCRIPPS RESEARCH INSTITUTE (US) 2010-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059179-A1 PALLADIUM-CATALYZED ORTHO-FLUORINATION POF1B, OCIAD2, ODC1 PTGS1 4856/4885PTGS2 4566/4885CA2 3314/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.