SCHEMBL14075554

SCHEMBL14075554

NS(=O)(=O)c1ccc(-c2ccno2)s1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 15/20 0.54
CA2 P00918 15/20 0.54
CA12 O43570 13/20 0.54
CA9 Q16790 13/20 0.54
CA4 P22748 2/20 0.50
CA7 P43166 2/20 0.50
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
FAAH O00519 1/20 0.38
PRF1 P14222 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2634053 0.83 CA1 (0.37) CA1CA2CA12CA9CA4
SCHEMBL788789 0.83 CA1 (0.37) CA1CA2CA12CA9CA4
SCHEMBL12319229 0.83 CA1 (0.40) CA1CA2CA12CA9CA4
SCHEMBL10154049 0.80 MAPT (0.44) CA1CA2CA12CA9NPC1
SCHEMBL15882624 0.80 MAPT (0.41) CA1CA2CA12CA9NPC1
SCHEMBL4802533 0.75 CA2 (0.53) CA1CA2CA12CA9CA4
SCHEMBL8747108 0.71 NPC1 (0.40) NPC1RAB9A
SCHEMBL29285931 0.69 MEN1 (0.66) NPC1RAB9APRF1
SCHEMBL1548721 0.68 POLB (0.52) CA1CA2CA12CA9CA4
SCHEMBL4109831 0.68 KDM4E (0.60) CA1CA2CA12CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026087527-A1 NOVEL TRPM4 ANTAGONISTS AND MEDICAL USE THEREOF Universitätsklinikum Hamburg-Eppendorf (DE) 2026-04-30 WO claimed
EP-4733298-A1 NOVEL TRPM4 ANTAGONISTS AND MEDICAL USE THEREOF Universitätsklinikum Hamburg-Eppendorf (DE) 2026-04-29 EP claimed
WO-2026087527-A1 NOVEL TRPM4 ANTAGONISTS AND MEDICAL USE THEREOF Universitätsklinikum Hamburg-Eppendorf (DE) 2026-04-30 WO disclosed
EP-4733298-A1 NOVEL TRPM4 ANTAGONISTS AND MEDICAL USE THEREOF Universitätsklinikum Hamburg-Eppendorf (DE) 2026-04-29 EP disclosed
US-7419962-B2 3,6-bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2008-09-02 US disclosed
US-7419962-B2 3,6-bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2008-09-02 US disclosed
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES ENANTA PHARMACEUTICALS, INC. 2008-01-31 US disclosed
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES ENANTA PHARMACEUTICALS, INC. 2008-01-31 US disclosed
WO-2008014221-A2 BRIDGED CARBAMATE MACROLIDES ENANTA PHARMACEUTICALS, INC. (US) 2008-01-31 WO disclosed
US-7312201-B2 Tetracyclic bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-12-25 US disclosed
US-7312201-B2 Tetracyclic bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-12-25 US disclosed
US-7291602-B2 11,12-lactone bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-11-06 US disclosed
US-7291602-B2 11,12-lactone bicyclolides ENANTA PHARMACEUTICALS, INC. (US) 2007-11-06 US disclosed
WO-2007115278-A2 3,6,11-TRICYCLOLIDE ENANTA PHARMACEUTICALS, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080027012-A1 BRIDGED CARBAMATE MACROLIDES HDAC6, SI, HDAC3 CA1 2023/4885CA2 363/4885CA12 378/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.