SCHEMBL14099804

SCHEMBL14099804

BCC(=O)N(Cc1ccccc1F)C1Cc2ccccc2C1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
C5AR1 P21730 1/20 0.46
OPRM1 P35372 2/20 0.45
ALDH1A1 P00352 9/20 0.43
THRB P10828 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
MC4R P32245 1/20 0.38
MC5R P33032 1/20 0.38
MC3R P41968 1/20 0.38
RIPK1 Q13546 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207029 0.88 C5AR1 (0.47) C5AR1OPRM1ALDH1A1THRBKDM4E
SCHEMBL6206609 0.86 C5AR1 (0.46) C5AR1OPRM1ALDH1A1THRBKDM4E
SCHEMBL5047630 0.78 ALDH1A1 (0.43) C5AR1OPRM1ALDH1A1THRBKDM4E
SCHEMBL5047628 0.78 C5AR1 (0.44) C5AR1OPRM1ALDH1A1THRBKDM4E
SCHEMBL5135947 0.75 MAPT (0.48) C5AR1OPRM1ALDH1A1KDM4EMAPT
SCHEMBL6342543 0.74 C5AR1 (0.56) C5AR1OPRM1ALDH1A1THRBMEN1
SCHEMBL5136013 0.74 C5AR1 (0.56) C5AR1OPRM1ALDH1A1THRBMEN1
SCHEMBL19002822 0.73 OPRM1 (0.69) OPRM1ALDH1A1THRBLMNAMEN1
SCHEMBL5134730 0.73 C5AR1 (0.57) C5AR1OPRM1ALDH1A1THRBMEN1
SCHEMBL5136309 0.73 C5AR1 (0.55) C5AR1OPRM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322309-B1 HIGH AFFINITY SMALL MOLECULE C5A RECEPTOR MODULATORS NEUROGEN CORP (US) 2008-08-13 EP disclosed