SCHEMBL14100577

SCHEMBL14100577

CBc1cc(C)cnc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.56
NOS2 P35228 4/20 0.56
NOS1 P29475 3/20 0.56
CYP2A6 P11509 2/20 0.40
CCR1 P32246 2/20 0.35
CCR5 P51681 2/20 0.35
CCR8 P51685 2/20 0.35
CYP1A2 P05177 1/20 0.32
KMT2A Q03164 2/20 0.31
HTT P42858 2/20 0.31
KDM4E B2RXH2 2/20 0.31
UHRF1 Q96T88 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
BLM P54132 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HSD17B10 Q99714 1/20 0.31
IKBKB O14920 1/20 0.31
XDH P47989 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13515059 0.77 IDO1 (0.39) NOS3NOS2NOS1CYP1A2KMT2A
SCHEMBL14100526 0.74 KDM4E (0.36) NOS3NOS2NOS1CCR1CCR5
SCHEMBL14100837 0.74 CCR1 (0.35) NOS3NOS2NOS1CCR1CCR5
SCHEMBL172774 0.72
SCHEMBL31619921 0.72
SCHEMBL91450 0.72
SCHEMBL24139999 0.71 NOS3 (0.33) NOS3NOS2NOS1CCR1CCR5
SCHEMBL118541 0.68
SCHEMBL29690486 0.68
SCHEMBL91444 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337251-B1 MONOCYCLIC OR BICYCLIC CARBOCYCLES AND HETEROCYCLES AS FACTOR XA INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2008-08-20 EP disclosed