SCHEMBL14101047

SCHEMBL14101047

CC(C)[C@]1(C(=O)N2CCc3ccc(-c4cccnc4)cc3C2)CCC(N)C1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 15/20 0.64
CYP11B1 P15538 4/20 0.47
CYP11B2 P19099 3/20 0.46
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14599192 1.00 CCR2 (0.64) CCR2CYP11B1CYP11B2KDM1A
SCHEMBL14629237 0.84 CCR2 (0.69) CCR2
SCHEMBL14101049 0.84 CCR2 (0.69) CCR2
SCHEMBL14101159 0.84 CCR2 (0.59) CCR2CYP11B1CYP11B2
SCHEMBL14599194 0.83 CCR2 (0.66) CCR2KDM1A
SCHEMBL13646017 0.82 CCR2 (0.59) CCR2CYP11B2
SCHEMBL14100872 0.78 CCR2 (0.58) CCR2
SCHEMBL5549022 0.77 CCR2 (0.70) CCR2
SCHEMBL14344815 0.77 CCR2 (0.70) CCR2
SCHEMBL14107452 0.74 CCR2 (0.49) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501803-B1 TETRAHYDROPYRANYL CYCLOPENTYL TETRAHYDROISOQUINOLINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2008-08-13 EP disclosed