SCHEMBL14101159

SCHEMBL14101159

CC(C)[C@]1(C(=O)N2CCc3ccc(-c4cccnc4)cc3C2)CCC(N(C)C2CCOCC2)C1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 18/20 0.59
CYP11B1 P15538 2/20 0.41
KCNH2 Q12809 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101049 0.85 CCR2 (0.69) CCR2
SCHEMBL14629237 0.85 CCR2 (0.69) CCR2
SCHEMBL14599192 0.84 CCR2 (0.64) CCR2CYP11B1CYP11B2
SCHEMBL14101047 0.84 CCR2 (0.64) CCR2CYP11B1CYP11B2
SCHEMBL14101162 0.83 CCR2 (0.54) CCR2KCNH2
SCHEMBL14100848 0.81 CCR2 (0.61) CCR2
SCHEMBL14101080 0.79 CCR2 (0.49) CCR2
SCHEMBL14101101 0.79 CCR2 (0.48) CCR2KCNH2
SCHEMBL14599194 0.76 CCR2 (0.66) CCR2
SCHEMBL13646017 0.76 CCR2 (0.59) CCR2KCNH2CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501803-B1 TETRAHYDROPYRANYL CYCLOPENTYL TETRAHYDROISOQUINOLINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2008-08-13 EP disclosed