SCHEMBL14101707

SCHEMBL14101707

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(N4CCCC4)ccc3C(F)(F)F)c(=O)c3c2CCCN3)c1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.33
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CRHBP P24387 1/20 0.31
CASP1 P29466 1/20 0.31
CYP2C19 P33261 1/20 0.31
CASP7 P55210 1/20 0.31
CRHR2 Q13324 1/20 0.31
NOTUM Q6P988 3/20 0.31
TNK1 Q13470 2/20 0.31
IMPDH2 P12268 2/20 0.31
LMNA P02545 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719078 0.91 PARP1 (0.30) PARP1MEN1KMT2ACYP1A2CRHBP
SCHEMBL4719220 0.91 P2RX7 (0.34)
SCHEMBL4719218 0.91 P2RX7 (0.34)
SCHEMBL4720122 0.91 P2RX7 (0.34)
SCHEMBL4721704 0.88 MEN1 (0.34) PARP1MEN1KMT2ACYP1A2CRHBP
SCHEMBL4721052 0.86 MEN1 (0.31) MEN1KMT2ACYP1A2CRHBPCASP1
SCHEMBL4723349 0.84 PTK2 (0.30)
SCHEMBL4719523 0.81 P2RX7 (0.34) MEN1KMT2ACYP1A2CRHBPCASP1
SCHEMBL4720197 0.80
SCHEMBL4720292 0.80 P2RX7 (0.36) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed