SCHEMBL14101912

SCHEMBL14101912

COc1cncc(-c2nn(-c3cc(N4CCCC4)ccc3C(F)(F)F)c(=O)c3[nH]ccc23)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
AR P10275 1/20 0.34
CYP1A2 P05177 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34
TUBB2B Q9BVA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722822 0.92 F2 (0.37) ARCYP1A2TUBB4ATUBBTUBA3C
SCHEMBL4722458 0.89 ABL1 (0.39) CYP11B1CYP11B2CHRNB2CHRNA4F10
SCHEMBL4722453 0.89 ABL1 (0.39) CYP11B1CYP11B2CHRNB2CHRNA4F10
SCHEMBL14102050 0.84 PDE10A (0.37) ARCYP1A2MAP4K1MAPTHTT
SCHEMBL4719947 0.81 BACE1 (0.33) MAPTHTTHTR6
SCHEMBL4724251 0.80 KHK (0.36) F10MAPTHTTHTR6MAPK1
SCHEMBL4718877 0.80 P2RX7 (0.35) F2F10
SCHEMBL4718873 0.80 P2RX7 (0.35) F2F10
SCHEMBL14101715 0.79 AR (0.38) ARTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL14101716 0.77 AR (0.36) ARTUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed