SCHEMBL4718877

SCHEMBL4718877

COc1cc(OC)cc(-c2nn(-c3cc(N4CCC(O)C4)ccc3C(F)(F)F)c(=O)c3[nH]ccc23)c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.35
PDE3B Q13370 3/20 0.35
PDE3A Q14432 3/20 0.35
PDE7A Q13946 1/20 0.35
ITGB2 P05107 2/20 0.35
ICAM1 P05362 2/20 0.35
ITGAL P20701 2/20 0.35
RORC P51449 1/20 0.34
SOS1 Q07889 2/20 0.34
ROCK2 O75116 1/20 0.33
F10 P00742 4/20 0.33
F2 P00734 1/20 0.33
HSD11B1 P28845 3/20 0.33
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718873 1.00 P2RX7 (0.35) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4722458 0.93 ABL1 (0.39) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4722453 0.93 ABL1 (0.39) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4724504 0.90 ITGB2 (0.38) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4724501 0.90 ITGB2 (0.38) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4719571 0.89 PDE7A (0.38) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4719565 0.89 PDE7A (0.38) P2RX7PDE3BPDE3APDE7AITGB2
SCHEMBL4723310 0.88 ITGB2 (0.40) ITGB2ICAM1ITGAL
SCHEMBL4723315 0.88 ITGB2 (0.40) ITGB2ICAM1ITGAL
SCHEMBL4722822 0.88 F2 (0.37) F10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed