SCHEMBL14110451

SCHEMBL14110451

O=C1COC(NC(=O)O[C@@H](CC2CCCCC2)C(=O)N2CCOCC2)C1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSS P25774 18/20 0.47
CTSL P07711 6/20 0.46
CTSK P43235 4/20 0.46
REN P00797 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CTSB P07858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12196292 0.82 CTSS (0.49) CTSSCTSLCTSKRENALDH1A1
SCHEMBL12196236 0.82 CTSS (0.49) CTSSCTSLCTSKRENALDH1A1
SCHEMBL8289701 0.81 CTSS (0.48) CTSSCTSLCTSKREN
SCHEMBL12196239 0.76 CTSS (0.47) CTSSCTSLCTSKRENALDH1A1
SCHEMBL2162740 0.76 CTSS (0.43) CTSSCTSLCTSKRENCTSB
SCHEMBL8290883 0.74 CTSS (0.48) CTSSCTSLCTSKRENALDH1A1
SCHEMBL12196312 0.74 CTSK (0.58) CTSSCTSLCTSK
SCHEMBL2163908 0.74 CTSK (0.58) CTSSCTSLCTSK
SCHEMBL12196307 0.73 CTSS (0.53) CTSSCTSLCTSKCTSB
SCHEMBL12196296 0.73 CTSS (0.56) CTSSCTSLCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1744755-B1 COMPOUNDS AND COMPOSITIONS AS CATHEPSIN S INHIBITORS IRM LLC (BM) 2012-12-05 EP claimed