SCHEMBL14136181

SCHEMBL14136181

CC(C)c1cc(NC(=O)CNc2ccc(Oc3ccncc3)cc2)no1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 4/20 0.50
RIPK2 O43353 1/20 0.50
ALDH1A1 P00352 5/20 0.46
MAPT P10636 2/20 0.46
KMT2A Q03164 1/20 0.46
NLRP1 Q9C000 1/20 0.46
GAA P10253 1/20 0.44
TP53 P04637 2/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
GRK2 P25098 4/20 0.41
ROCK2 O75116 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
NPY5R Q15761 1/20 0.40
GALR3 O60755 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4444438 0.83 RAF1 (0.72) RAF1RIPK2
SCHEMBL13972318 0.83 RAF1 (0.48) RAF1RIPK2ALDH1A1MAPTKMT2A
SCHEMBL4441367 0.78 RAF1 (0.73) RAF1RIPK2ALDH1A1MAPTKMT2A
SCHEMBL13823410 0.78 RAF1 (0.50) RAF1RIPK2ALDH1A1MAPTKMT2A
SCHEMBL4443071 0.74 RAF1 (0.61) RAF1RIPK2GRK2GRK3
SCHEMBL13815845 0.73 RAF1 (0.72) RAF1RIPK2KMT2ANPC1RAB9A
SCHEMBL13823425 0.73 GRK2 (0.53) RAF1RIPK2LMNAGRK2ROCK2
SCHEMBL937763 0.69 RAF1 (0.70) RAF1RIPK2ALDH1A1LMNA
SCHEMBL4442571 0.69 RAF1 (0.62) RAF1RIPK2GRK2ROCK2GRK3
SCHEMBL4445772 0.68 CDK8 (0.56) RAF1RIPK2ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531817-B1 GLYCINAMIDE DERIVATIVES AS RAF-KINASE INHIBITORS MERCK PATENT GMBH (DE) 2008-07-30 EP disclosed