SCHEMBL14136367

SCHEMBL14136367

CN1CCN(c2nc(C(F)(F)F)nc3ccccc23)CC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 2/20 0.76
CYP1A2 P05177 3/20 0.65
CYP3A4 P08684 3/20 0.65
CYP2D6 P10635 2/20 0.65
MAPK1 P28482 2/20 0.65
HTR3E A5X5Y0 2/20 0.64
HTR3B O95264 2/20 0.64
HTR3A P46098 2/20 0.64
HTR3D Q70Z44 2/20 0.64
HTR3C Q8WXA8 2/20 0.64
HRH4 Q9H3N8 3/20 0.63
ALDH1A1 P00352 3/20 0.60
KDM4E B2RXH2 2/20 0.60
CCNE2 O96020 1/20 0.58
CCNE1 P24864 1/20 0.58
CDK2 P24941 1/20 0.58
TSHR P16473 2/20 0.56
LMNA P02545 2/20 0.56
HSD17B10 Q99714 1/20 0.56
HTR6 P50406 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23657801 0.83 TLR7 (0.72) TLR7CYP1A2CYP3A4CYP2D6MAPK1
SCHEMBL2710555 0.83 TLR7 (0.76) TLR7CYP1A2CYP3A4CYP2D6ALDH1A1
SCHEMBL4085139 0.79 RAB9A (0.78) CYP1A2CYP3A4CYP2D6MAPK1HRH4
SCHEMBL5320912 0.78 HTR3B (0.69) CYP1A2CYP3A4CYP2D6MAPK1HTR3E
SCHEMBL13125713 0.78 HRH4 (1.00) CYP1A2CYP3A4CYP2D6MAPK1HTR3E
Hydrochloric Acid SCHEMBL11740107 0.77 HTR3B (0.68) CYP1A2CYP3A4CYP2D6MAPK1HTR3E
SCHEMBL6125247 0.77 TSHR (0.84) CYP1A2CYP3A4CYP2D6MAPK1HTR3E
SCHEMBL4085081 0.75 HTR3E (0.66) CYP1A2CYP3A4CYP2D6MAPK1HTR3E
SCHEMBL27866870 0.75 HTR3E (0.66) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL15963530 0.75 TLR7 (0.59) TLR7CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1950199-A1 Proline derivatives and use thereof as drugs Mitsubishi Tanabe Pharma Corporation (JP) 2008-07-30 EP disclosed
EP-1930319-A1 Proline derivatives and use thereof as drugs Mitsubishi Tanabe Pharma Corporation (JP) 2008-06-11 EP disclosed