SCHEMBL14153754

SCHEMBL14153754

c1ccc(-c2ccc(-c3nc4c([nH]3)CCCC4)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
NPY5R Q15761 6/20 0.51
SMPD3 Q9NY59 1/20 0.49
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
TNKS O95271 1/20 0.41
PARP1 P09874 1/20 0.41
WNT3A P56704 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
MAPK13 O15264 1/20 0.41
RAF1 P04049 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861541 0.96 KMT2A (0.57) KMT2AL3MBTL1NPY5RSMPD3KDM4E
SCHEMBL15913449 0.86 KMT2A (0.44) KMT2AL3MBTL1NPY5RSMPD3KDM4E
SCHEMBL25220187 0.83 SMPD3 (0.49) KMT2AL3MBTL1NPY5RSMPD3KDM4E
SCHEMBL14153752 0.83 SMPD3 (0.49) KMT2AL3MBTL1NPY5RSMPD3KDM4E
SCHEMBL11844688 0.79 TNKS2 (0.50) KMT2AL3MBTL1SMPD3TNKSPARP1
SCHEMBL8319716 0.75 PDCD1 (0.53) KMT2AL3MBTL1NPY5RKDM4EALDH1A1
SCHEMBL12492799 0.75 PDCD1 (0.68) KMT2AL3MBTL1NPY5RKDM4EALDH1A1
SCHEMBL25120538 0.73 NPY5R (0.39) KMT2AL3MBTL1NPY5RSMPD3KDM4E
SCHEMBL22408471 0.73 ALDH1A1 (0.49) L3MBTL1NPY5RSMPD3KDM4EALDH1A1
SCHEMBL1032502 0.73 TNKS2 (0.68) KMT2AL3MBTL1KDM4EALDH1A1TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012162635-A1 METABOTROPIC GLUTAMATE RECEPTORS 5 MODULATORS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2012-11-29 WO disclosed