SCHEMBL1415499

SCHEMBL1415499

CC(C)C(CCC(=O)NC(COC(C)(C)C)c1nnnn1Cc1ccccc1)NCc1cc(Oc2ccccc2)ncc1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 19/20 0.40
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1413920 1.00 GHSR (0.40) GHSRHDAC1HDAC6
SCHEMBL1414565 0.90 GHSR (0.43) GHSRHDAC1HDAC6
SCHEMBL4038449 0.77 PIN1 (0.36)
SCHEMBL4038445 0.77 PIN1 (0.36)
SCHEMBL1414241 0.77 S1PR1 (0.37)
SCHEMBL1414468 0.77 S1PR1 (0.37)
SCHEMBL1414469 0.77 S1PR1 (0.37)
SCHEMBL1414267 0.76 GHSR (0.51) GHSRHDAC1HDAC6
SCHEMBL1414271 0.76 GHSR (0.51) GHSRHDAC1HDAC6
SCHEMBL1414214 0.74 GHSR (0.41) GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966198-B1 2-AMINO-3,4-DIHYDRO-PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) JANSSEN PHARMACEUTICA NV (BE) 2011-03-16 EP disclosed