SCHEMBL1415951

SCHEMBL1415951

CC(=O)N(N)C(=O)c1ccncc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
KMT2A Q03164 2/20 0.49
NAPRT Q6XQN6 1/20 0.45
TP53 P04637 1/20 0.44
MPO P05164 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.41
HSD17B10 Q99714 2/20 0.41
MLYCD O95822 1/20 0.40
ALOX15 P16050 1/20 0.40
GAA P10253 1/20 0.38
LTA4H P09960 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6503060 0.87 NAPRT (0.52) KDM4EKMT2ANAPRTTP53MPO
SCHEMBL2988329 0.83 NAPRT (0.48) KDM4EKMT2ANAPRTTP53MPO
SCHEMBL7554003 0.83 KMT2A (0.45) KDM4EKMT2ANAPRTMPOCYP1A2
SCHEMBL7554228 0.80 KMT2A (0.42) KDM4EKMT2ANAPRTTP53MPO
SCHEMBL3935110 0.80 NAPRT (0.45) KDM4EKMT2ANAPRTMPOCYP1A2
SCHEMBL6614684 0.80 NAPRT (0.45) KDM4EKMT2ANAPRTMPOCYP1A2
SCHEMBL21805934 0.79 KDM4E (0.45) KDM4EKMT2ANAPRTTP53MPO
SCHEMBL7584545 0.79 KDM4E (0.44) KDM4EKMT2ANAPRTMPOCYP1A2
SCHEMBL11590778 0.79 KDM4E (0.56) KDM4EKMT2ANAPRTTP53MPO
SCHEMBL5452316 0.79 CES2 (0.46) NAPRTCYP3A4CYP2C19LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170101678-A1 METHOD FOR SCREENING RISK OF DRUG-INDUCED TOXICITY RESEARCH CENTER FOR BIOTECHNOLOGY AND MEDICINE POLICY (TW) 2017-04-13 US disclosed
CN-105940116-A Method for screening risk of drug-induced toxicity 财团法人生技医疗科技政策研究中心 2016-09-14 CN disclosed
WO-2015109608-A1 METHOD FOR SCREENING RISK OF DRUG-INDUCED TOXICITY 财团法人生技医疗科技政策研究中心 2015-07-30 WO disclosed
US-8577617-B2 Metabolic phenotyping CLAYTON THOMAS ANDREW (GB) 2013-11-05 US disclosed
EP-1540560-B1 METABOLIC PHENOTYPING PFIZER LTD (GB) 2011-03-16 EP disclosed
US-20100184811-A1 ISONIAZID MEDIATED HEALING OF WOUNDS AND ULCERS BRIDGE BIORESEARCH RIGHTS (JERSEY) LIMITED (GB) 2010-07-22 US disclosed
WO-2010037134-A2 MULTI-STAGE STEM CELL CARCINOGENESIS STEMLIFELINE, INC. (US) 2010-04-01 WO disclosed
US-20090192721-A1 METABOLIC PHENOTYPING PFIZER INC 2009-07-30 US disclosed
EP-1540560-A2 METABOLIC PHENOTYPING Pfizer Limited (GB) 2005-06-15 EP disclosed
US-20050074745-A1 Metabolic phenotyping PFIZER INC 2005-04-07 US disclosed
WO-2003107270-A2 METABOLIC PHENOTYPING PFIZER LIMITED (GB) 2003-12-24 WO disclosed
WO-2002043668-A2 ANTIMYCOBACTERIAL COMPOUNDS AND METHOD FOR MAKING THE SAME WELLESLEY COLLEGE (US) 2002-06-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100184811-A1 ISONIAZID MEDIATED HEALING OF WOUNDS AND ULCERS ODC1, OTC, ACACB KDM4E 3169/4885KMT2A 4030/4885NAPRT 246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.