SCHEMBL6503060

SCHEMBL6503060

NN(C(=O)c1ccncc1)C(=O)c1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.52
KDM4E B2RXH2 3/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C19 P33261 2/20 0.50
MPO P05164 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CYP2A6 P11509 1/20 0.50
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.46
LMNA P02545 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 1/20 0.43
LTA4H P09960 1/20 0.43
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
HTT P42858 1/20 0.42
PLOD2 O00469 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2988329 0.91 NAPRT (0.48) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL6614684 0.87 NAPRT (0.45) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL1415951 0.87 KDM4E (0.49) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL3935110 0.87 NAPRT (0.45) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL27810441 0.86 NAPRT (0.52) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL21144262 0.84 CA1 (0.43) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL21805934 0.82 KDM4E (0.45) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL7584545 0.82 KDM4E (0.44) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL7554003 0.82 KMT2A (0.45) NAPRTKDM4EKMT2ACYP1A2CYP3A4
SCHEMBL1527753 0.82 CES2 (0.47) NAPRTKDM4EKMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6846933-B1 Antimycobacterial compounds and method for making the same THE BOARD OF TRUSTEES OF WELLESLEY COLLEGE (US) 2005-01-25 US disclosed
WO-2002043668-A2 ANTIMYCOBACTERIAL COMPOUNDS AND METHOD FOR MAKING THE SAME WELLESLEY COLLEGE (US) 2002-06-06 WO disclosed