SCHEMBL14178552

SCHEMBL14178552

CC(C)CCN(C)Cc1ccc2oc3ccc(C(N)=O)cc3c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
HTR1D P28221 2/20 0.43
HTR2C P28335 2/20 0.43
F2 P00734 2/20 0.39
F10 P00742 2/20 0.39
F7 P08709 2/20 0.39
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
OPRM1 P35372 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14369641 0.80 OPRM1 (0.39) HTR1AHTR1DHTR2CF2F10
SCHEMBL4965627 0.78 OPRM1 (0.50) HTR1AHTR1DHTR2CNPSR1OPRM1
Trifluoroacetic Acid SCHEMBL4967345 0.74 TRPM8 (0.37) HTR1AHTR1DHTR2CF2F10
SCHEMBL1346996 0.74 TRPV1 (0.49) RORC
SCHEMBL3691407 0.71 LPAR1 (0.53) BCHEACHEOPRM1SLC6A2SLC6A4
SCHEMBL14369647 0.70 HIF1A (0.33) F2F10F7BCHEACHE
SCHEMBL14369648 0.70 F2 (0.34) F2F10F7OPRM1TSHR
SCHEMBL4984818 0.70 MRGPRX4 (0.49) KDM4EALDH1A1LMNA
SCHEMBL3699746 0.68 OPRM1 (0.43) BCHEACHEOPRM1SLC6A2SLC6A3
SCHEMBL21864736 0.67 GSK3B (0.40) KDM4EALDH1A1LMNAL3MBTL1IKBKE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP disclosed