SCHEMBL14181791

SCHEMBL14181791

CC(C)(C)OC(=O)NC(Cc1ccc2c(c1)NC(=O)C(CCC1NC(=N)NC1=O)O2)C(=O)OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.40
CCKAR P32238 1/20 0.40
CCKBR P32239 1/20 0.40
CTSK P43235 3/20 0.39
CTSL P07711 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
EPHX2 P34913 1/20 0.38
TACR1 P25103 1/20 0.38
KLK5 Q9Y337 2/20 0.38
KLK7 P49862 1/20 0.37
PPARA Q07869 1/20 0.37
TDO2 P48775 1/20 0.37
ACE P12821 1/20 0.37
CTSS P25774 2/20 0.36
PSMB1 P20618 1/20 0.36
PSMB8 P28062 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3049757 0.90 IDO1 (0.44) IDO1CCKARCCKBRCTSKPPARA
SCHEMBL7160937 0.86 IDO1 (0.43) IDO1CCKARCCKBRCTSKPPARA
SCHEMBL7363237 0.86 CCKAR (0.44) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL7363235 0.83 KLK5 (0.42) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL7166021 0.82 ACE (0.47) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL7469657 0.81 MAPT (0.44) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL7163527 0.80 MAPT (0.46) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL7372914 0.80 HSD17B10 (0.41) IDO1CCKARCCKBRCTSKCTSL
SCHEMBL8330384 0.79 IDO1 (0.40) IDO1CCKARCCKBRCTSKPOLB
SCHEMBL4683912 0.79 IDO1 (0.40) IDO1CCKARCCKBRCTSKPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7371854-B2 Method for the production of bicyclic aromatic amino acids and intermediate products thereof MERCK PATENT GMBH (DE) 2008-05-13 US disclosed
US-7371854-B2 Method for the production of bicyclic aromatic amino acids and intermediate products thereof MERCK PATENT GMBH (DE) 2008-05-13 US disclosed