SCHEMBL8330384

SCHEMBL8330384

CCOC(=O)[C@H](Cc1ccc2c(c1)NC(=O)C(CCC(=O)O)O2)NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.40
CCKAR P32238 1/20 0.40
CCKBR P32239 1/20 0.40
USP2 O75604 1/20 0.39
GAA P10253 1/20 0.39
SCN9A Q15858 1/20 0.39
ACE P12821 1/20 0.38
EPHX2 P34913 1/20 0.38
HSD17B10 Q99714 2/20 0.38
KLK5 Q9Y337 1/20 0.38
ALOX15 P16050 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4683912 1.00 IDO1 (0.40) IDO1CCKARCCKBRUSP2GAA
SCHEMBL7167872 0.91 IDO1 (0.46) IDO1CCKARCCKBRUSP2GAA
SCHEMBL4680395 0.91 USP2 (0.39) USP2GAAHSD17B10ALOX15L3MBTL1
SCHEMBL4679583 0.91 USP2 (0.39) USP2GAAHSD17B10ALOX15L3MBTL1
SCHEMBL7363235 0.90 KLK5 (0.42) IDO1CCKARCCKBRUSP2GAA
SCHEMBL4685497 0.88 USP2 (0.37) IDO1CCKARCCKBRUSP2GAA
SCHEMBL4850590 0.85 CCKAR (0.35) CCKARCCKBRUSP2GAASCN9A
SCHEMBL7469657 0.85 MAPT (0.44) IDO1CCKARCCKBRHSD17B10KLK5
SCHEMBL8326662 0.84 USP2 (0.37) USP2GAAHSD17B10ALOX15L3MBTL1
SCHEMBL4680620 0.83 ITGB3 (0.43) IDO1USP2GAAACEHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7371854-B2 Method for the production of bicyclic aromatic amino acids and intermediate products thereof MERCK PATENT GMBH (DE) 2008-05-13 US disclosed
US-7371854-B2 Method for the production of bicyclic aromatic amino acids and intermediate products thereof MERCK PATENT GMBH (DE) 2008-05-13 US disclosed
WO-2004072054-A1 METHOD FOR THE PRODUCTION OF BICYCLIC AROMATIC AMINO ACIDS AND INTERMEDIATE PRODUCTS THEREOF MERCK PATENT GMBH (DE) 2004-08-26 WO disclosed