SCHEMBL14190089

SCHEMBL14190089

CC(=O)NC(C(=O)OCc1cc(C(O)CNC(C)(C)C)ccc1O)C(C)(C)SC(=O)CCCO[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 6/20 0.42
CYP2D6 P10635 3/20 0.42
ADRB1 P08588 2/20 0.42
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
HIF1A Q16665 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
PMP22 Q01453 1/20 0.41
ADRB3 P13945 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
KCNH2 Q12809 1/20 0.33
LMNA P02545 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2966767 0.83 ADRB2 (0.51) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL14117385 0.80 ADRB2 (0.49) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL1230900 0.77 ADRB2 (0.63) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL12158793 0.73 ADRB2 (0.66) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL6838978 0.73 ADRB2 (0.66) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL13240114 0.70 ADRB2 (0.42) ADRB2ADRB1ADRB3
SCHEMBL14141543 0.68 ADRB2 (0.62) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL7778381 0.68 ADRB2 (0.56) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL5145221 0.68 ADRB2 (0.56) ADRB2CYP2D6ADRB1CYP1A2TSHR
SCHEMBL7775809 0.68 ADRB2 (0.56) ADRB2CYP2D6ADRB1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378412-B2 Pharmaceutical compounds NICOX S.A. (FR) 2008-05-27 US disclosed