SCHEMBL1419785

SCHEMBL1419785

CC(C)(C)OC(=O)[AsH]c1cccc(COS(C)(=O)=O)n1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
PTGER2 P43116 1/20 0.32
ALOX5 P09917 1/20 0.31
NQO2 P16083 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL465906 0.75 CCR2 (0.43) PTGER2NQO2
SCHEMBL25321212 0.74 KCNH2 (0.44) CYP1A2CYP3A4CYP2D6
SCHEMBL945801 0.73 CYP1A2 (0.36) CYP1A2CYP3A4CYP2D6PTGER2NQO2
SCHEMBL24915330 0.72 HCRTR1 (0.40) CYP1A2CYP3A4CYP2D6
SCHEMBL9902359 0.71 CYP1A2 (0.33) CYP1A2CYP3A4CYP2D6PTGER2NQO2
SCHEMBL17247586 0.70 CYP1A2 (0.40) CYP1A2CYP3A4CYP2D6
SCHEMBL17963027 0.70 CYP1A2 (0.44) CYP1A2CYP3A4CYP2D6
SCHEMBL4714316 0.69 CYP1A2 (0.35) CYP1A2CYP3A4CYP2D6
SCHEMBL4470267 0.69 MEN1 (0.39) CYP1A2CYP3A4CYP2D6
SCHEMBL1556569 0.69 GPR119 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297144-A1 IMIDAZOPYRIDINE AND RELATED ANALOGS AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2011-03-23 EP disclosed
WO-2009146358-A1 IMIDAZOPYRIDINE AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2009-12-03 WO disclosed