SCHEMBL14199040

SCHEMBL14199040

Cc1cc2ncccc2cc1C(F)(F)c1nnc2ccc(-c3cccc(N)c3)nn12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 18/20 0.58
PDE3B Q13370 2/20 0.52
PDE3A Q14432 2/20 0.52
NQO2 P16083 1/20 0.52
PIP4K2C Q8TBX8 1/20 0.52
PDE1A P54750 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
PDE1C Q14123 1/20 0.43
PDE11A Q9HCR9 1/20 0.43
PDE10A Q9Y233 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GABRA1 P14867 1/20 0.41
HPGD P15428 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12049504 0.87 MET (0.57) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL14199066 0.81 MET (0.67) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL12049507 0.80 MET (0.67) MET
SCHEMBL14198917 0.78 MET (0.54) METPDE3BPDE3APDE1APDE4C
SCHEMBL14198919 0.78 MET (0.54) MET
SCHEMBL14199047 0.77 MET (0.52) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL12049503 0.74 MET (0.81) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL12049487 0.74 MET (0.81) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL12049490 0.74 MET (0.84) METPDE3BPDE3ANQO2PIP4K2C
SCHEMBL2496429 0.74 MET (0.76) METPDE3BPDE3ANQO2PIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051805-A2 TRIAZOLO-PYRIDAZINE PROTEIN KINASE MODULATORS SGX PHARMACEUTICALS, INC. (US) 2008-05-02 WO disclosed