SCHEMBL14199352

SCHEMBL14199352

O=CCn1c(=O)[nH]c2c(C(F)(F)F)cccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.37
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36
TLR7 Q9NYK1 2/20 0.36
KIF11 P52732 1/20 0.36
CHRM1 P11229 1/20 0.35
DAO P14920 3/20 0.35
HTR6 P50406 2/20 0.34
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34
GRIN1 Q05586 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14198905 0.75 DAO (0.42) SMN1; SMN2MEN1ALDH1A1LMNAHPGD
SCHEMBL12794217 0.71 POLB (0.51) KDM4ESMN1; SMN2MEN1ALDH1A1LMNA
SCHEMBL14198908 0.70 CYP1A2 (0.64) SMN1; SMN2MEN1ALDH1A1LMNAPOLB
SCHEMBL8344975 0.69 GRIA1 (0.55) MEN1KMT2AGRIN1GRIN2B
SCHEMBL31285844 0.66 CHRM1 (0.52) LMNAHTTCHRM1
SCHEMBL22605450 0.66 CHRM1 (0.52) LMNAHTTCHRM1
SCHEMBL22612923 0.63 EPHX2 (0.63) SMN1; SMN2MEN1ALDH1A1LMNAHPGD
SCHEMBL14518261 0.63 DAO (0.55) KDM4EMEN1KMT2ADAO
SCHEMBL14198898 0.63 DAO (0.55) SMN1; SMN2KMT2AHSD17B10TLR7DAO
SCHEMBL3858995 0.62 HTR6 (0.53) KDM4ESMN1; SMN2ALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-B1 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-05-07 EP disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed