SCHEMBL14199540

SCHEMBL14199540

CC(F)(c1ccc2ncsc2c1)c1nnc2ccc(-c3cccc(N)c3)nn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 10/20 0.44
CYP1A2 P05177 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
GABRA1 P14867 1/20 0.41
HPGD P15428 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NQO2 P16083 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
PIP4K2C Q8TBX8 1/20 0.40
FYN P06241 2/20 0.40
PFKFB3 Q16875 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12049429 0.90 MET (0.45) METCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL12049427 0.88 MET (0.46) METCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL14199066 0.83 MET (0.67) METNQO2PDE3BPDE3APIP4K2C
SCHEMBL12049426 0.79 MET (0.56) MET
SCHEMBL14205065 0.76 MET (0.52) METKDM4ECYP3A4HSD17B10NQO2
SCHEMBL14198923 0.76 MET (0.55) METPDE3BPDE3AFYNPFKFB3
SCHEMBL14198934 0.76 MET (0.55) METPDE3BPDE3AFYNPFKFB3
SCHEMBL14198933 0.76 MET (0.55) METPDE3BPDE3AFYNPFKFB3
SCHEMBL14198928 0.76 MET (0.60) MET
SCHEMBL12049397 0.72 MET (0.68) METNQO2PDE3BPDE3APIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051805-A2 TRIAZOLO-PYRIDAZINE PROTEIN KINASE MODULATORS SGX PHARMACEUTICALS, INC. (US) 2008-05-02 WO disclosed