SCHEMBL14199698

SCHEMBL14199698

C=C/C=c1/c(S(N)(=O)=O)ccc/c1=C/N

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.37
CA1 P00915 8/20 0.37
CA9 Q16790 7/20 0.37
CA6 P23280 3/20 0.36
CA12 O43570 3/20 0.36
CA4 P22748 2/20 0.36
CA5A P35218 2/20 0.36
CA7 P43166 2/20 0.36
CA5B Q9Y2D0 2/20 0.36
CYP2C9 P11712 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CDK2 P24941 1/20 0.36
MAPK1 P28482 1/20 0.33
STAT3 P40763 1/20 0.33
PTGES2 Q9H7Z7 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200446 0.77 CYP3A4 (0.46) CYP2C9MAPK1
SCHEMBL13038588 0.75 CYP3A4 (0.43) CYP2C9MAPK1
SCHEMBL8346103 0.72 CD44 (0.30)
SCHEMBL14199699 0.71
SCHEMBL16152376 0.65 ALDH1A1 (0.31)
SCHEMBL14199960 0.63 HTR1B (0.43) MAPK1
SCHEMBL202947 0.61 CA2 (0.70) CA2CA1CA9CA6CA12
SCHEMBL1142906 0.61 CA2 (0.50) CA2CA1CA9CA6CA12
SCHEMBL10077289 0.61 CD44 (0.30)
SCHEMBL9138970 0.60 CDK2 (0.78) CA2CA1CA9CA6CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284734-B1 ISOQUINOLINE DERIVATIVES AS PROTEIN KINASE INHIBITORS CUREGENICS LTD (IL) 2008-05-21 EP disclosed