SCHEMBL14200523

SCHEMBL14200523

Cc1cc(Cl)cc(-c2nnn(-c3ccccn3)n2)c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 14/20 0.53
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
NFKB1 P19838 1/20 0.42
CASP3 P42574 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698325 0.85 GRM5 (0.53) GRM5NPC1RAB9AMAPTPKM
SCHEMBL4698743 0.83 GRM5 (0.67) GRM5NPC1RAB9AMAPTPKM
SCHEMBL13683903 0.82 GRM5 (0.46) GRM5NPC1RAB9AMAPT
SCHEMBL4699888 0.81 GRM5 (0.72) GRM5
SCHEMBL4701228 0.81 GRM5 (0.72) GRM5
SCHEMBL13683938 0.81 GRM5 (0.53) GRM5NPC1RAB9AMAPTALDH1A1
SCHEMBL13683904 0.78 GRM5 (0.57) GRM5NPC1RAB9AMAPTPKM
SCHEMBL4700359 0.76 GRM5 (0.54) GRM5NPC1RAB9AMAPTALDH1A1
SCHEMBL13684502 0.76 GRM5 (0.45) GRM5NPC1RAB9AMAPTPKM
SCHEMBL13683939 0.72 GRM5 (0.54) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1434773-B1 HETEROARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK & CO INC (US) 2008-05-21 EP disclosed