SCHEMBL14201033

SCHEMBL14201033

CCC(CC)N(C(=O)CC(C)(C)C)c1ccc(F)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 8/20 0.33
RIPK1 Q13546 3/20 0.33
NPSR1 Q6W5P4 2/20 0.33
TSHR P16473 2/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
KDM4E B2RXH2 2/20 0.33
TDO2 P48775 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229578 0.90 RIPK1 (0.34) IDO1RIPK1NPSR1TSHRLMNA
SCHEMBL14201013 0.90 CYP1A2 (0.34) IDO1RIPK1NPSR1CYP1A2CYP2D6
SCHEMBL14201017 0.90 CYP1A2 (0.34) IDO1RIPK1NPSR1CYP1A2CYP2D6
SCHEMBL14201039 0.88 IDO1 (0.33) IDO1RIPK1NPSR1CYP1A2CYP2D6
SCHEMBL14200734 0.85 RIPK1 (0.34) RIPK1CYP1A2CYP2C19
SCHEMBL14200498 0.85 RIPK1 (0.39) RIPK1HDAC8
SCHEMBL14200858 0.85 CYP1A2 (0.33) IDO1RIPK1NPSR1CYP1A2CYP2D6
SCHEMBL14200486 0.84 ALDH1A1 (0.44) TSHRLMNAKDM4EALDH1A1
SCHEMBL14229460 0.84 NPSR1 (0.37) IDO1NPSR1TSHRLMNACYP1A2
SCHEMBL14201008 0.83 CHRNA1 (0.37) TSHRLMNACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed