SCHEMBL14201100

SCHEMBL14201100

O=C1c2ccccc2C(=O)c2c(NC(=O)c3ccc4c5c(nsc35)-c3ccccc3C4=O)cccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.49
CYP1A2 P05177 3/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 2/20 0.41
EGFR P00533 1/20 0.41
PABPC1 P11940 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CASP3 P42574 2/20 0.41
ALDH1A1 P00352 2/20 0.40
POLB P06746 2/20 0.40
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
DNMT1 P26358 1/20 0.40
RAD52 P43351 1/20 0.40
SMARCA2 P51531 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200817 1.00 MAOA (0.49) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200950 0.94 ADORA2A (0.44) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200962 0.93 CYP1A2 (0.45) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200811 0.93 CASP3 (0.43) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200944 0.90 MAOA (0.41) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200924 0.86 KDM4E (0.38) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200946 0.84 MAPT (0.43) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200867 0.84 MAPT (0.38) MAOACYP1A2MAPTKDM4EMAPK1
SCHEMBL14200935 0.84 POLB (0.48) MAOACYP1A2MAPTKDM4ESMN1; SMN2
SCHEMBL14200933 0.80 MAPT (0.46) CYP1A2MAPTKDM4EMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7354947-B2 Isothiazoloanthrones, isoxazoloanthrones, isoindolanthrones and derivatives thereof a JNK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC (US) 2008-04-08 US disclosed
US-7354947-B2 Isothiazoloanthrones, isoxazoloanthrones, isoindolanthrones and derivatives thereof a JNK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC (US) 2008-04-08 US disclosed