SCHEMBL14201833

SCHEMBL14201833

C[C@H](CN(C)C)[C@@](C)(O)c1cccc(ON)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP2C19 P33261 1/20 0.48
HSD17B10 Q99714 1/20 0.48
HIF1A Q16665 2/20 0.38
CYP3A4 P08684 2/20 0.38
MEN1 O00255 1/20 0.37
TTR P02766 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNH2 Q12809 3/20 0.37
SLC6A4 P31645 3/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.37
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
MRGPRX2 Q96LB1 1/20 0.36
CHRM3 P20309 1/20 0.36
HRH2 P25021 1/20 0.36
HTR2A P28223 1/20 0.36
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL355959 0.87 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
SCHEMBL169116 0.87 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
SCHEMBL8529142 0.87 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
Hydrochloric Acid SCHEMBL8686514 0.86 CYP2D6 (0.48) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
SCHEMBL13823445 0.84 CYP2D6 (0.46) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
SCHEMBL13823400 0.84 CYP2D6 (0.46) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A
SCHEMBL150354 0.80 ALDH1A1 (0.53) CYP2D6ALDH1A1CYP2C19HSD17B10CYP3A4
SCHEMBL150355 0.80 ALDH1A1 (0.53) CYP2D6ALDH1A1CYP2C19HSD17B10CYP3A4
SCHEMBL3730504 0.80 ALDH1A1 (0.53) CYP2D6ALDH1A1CYP2C19HSD17B10CYP3A4
Hydrochloric Acid SCHEMBL7673735 0.78 ALDH1A1 (0.51) CYP2D6ALDH1A1CYP2C19HSD17B10HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1509216-B1 ACTIVE INGREDIENT SALTS AND ESTERS OF 1-DIMETHYLAMINO-3-(3-METHOXY-PHENYL)-2-METHYL-PENTAN-3-OL AND 3-(3-DIMETHYLAMINO-1-ETHYL-1-HYDROXY-2-METHYL-PROPYL)-PHENOL GRUENENTHAL GMBH (DE) 2008-05-07 EP disclosed