SCHEMBL14212430

SCHEMBL14212430

O=c1n(Cc2ccc(C(F)(F)F)nc2)nc2c(-c3cccnc3)c(-c3ccc(Cl)cc3)cnn12

nearest known ligand 0.82

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.82
CYP2C9 P11712 5/20 0.52
CYP2C19 P33261 5/20 0.52
CYP3A4 P08684 4/20 0.52
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
NR3C1 P04150 1/20 0.38
PSD A5PKW4 2/20 0.36
GPR119 Q8TDV5 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14211170 0.92 CNR1 (0.86) CNR1CYP2C9CYP2C19CYP3A4PTGS2
SCHEMBL14181226 0.92 CNR1 (0.69) CNR1CYP2C9CYP2C19CYP3A4PTGS1
SCHEMBL14211173 0.91 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4PTGS1
SCHEMBL14211892 0.91 CNR1 (0.91) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14210241 0.91 CNR1 (0.84) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL4798385 0.91 CNR1 (1.00) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14181126 0.90 CNR1 (0.68) CNR1CYP2C9CYP2C19CYP3A4PTGS1
SCHEMBL14212431 0.89 CNR1 (0.78) CNR1CYP2C9CYP2C19CYP3A4PTGS2
SCHEMBL14211052 0.89 CNR1 (0.81) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14210240 0.89 CNR1 (0.81) CNR1CYP2C9CYP2C19CYP3A4NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378418-B2 Azabicyclic heterocycles as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed
EP-1697370-B1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-04-25 EP disclosed