SCHEMBL14213262

SCHEMBL14213262

C=C(C)Cc1cc(C)c(O)c(Cc2cc(CC(=C)C)cc(Cc3cc(CC(=C)C)cc(Cc4cc(CC(=C)C)cc(CC)c4O)c3O)c2O)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SHBG P04278 1/20 0.45
HSPA5 P11021 2/20 0.38
HMGB1 P09429 1/20 0.36
CXCL12 P48061 1/20 0.36
DHFR P00374 2/20 0.35
AMY1A P0DUB6 1/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
ALOX5 P09917 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
ESR1 P03372 2/20 0.30
ESR2 Q92731 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10046767 0.94 SHBG (0.46) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL14213248 0.91 SHBG (0.38) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL10046744 0.91 SHBG (0.38) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL7591262 0.83 SHBG (0.53) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL30003742 0.80 SHBG (0.63) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL2384360 0.80 SHBG (0.63) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL9405316 0.79 CA1 (0.44) SHBGHMGB1CXCL12CYP2C9ALOX5
SCHEMBL12998649 0.77 SHBG (0.59) SHBGHSPA5HMGB1CXCL12AMY1A
SCHEMBL69627 0.77 SHBG (0.70) SHBGHSPA5HMGB1CXCL12DHFR
SCHEMBL20102186 0.77 SHBG (0.55) SHBGHSPA5HMGB1CXCL12DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8716343-B2 Calixarene-based peptide conformation mimetics, methods of use, and methods of making REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2014-05-06 US disclosed
US-8642656-B2 Calixarene-based peptide conformation mimetics, methods of use, and methods of making REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2014-02-04 US disclosed
US-20130035394-A1 Calixarene-Based Peptide Conformation Mimetics, Methods of Use, and Methods of Making REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2013-02-07 US disclosed
US-20120309801-A1 CALIXARENE-BASED PEPTIDE CONFORMATION MIMETICS, METHODS OF USE, AND METHODS OF MAKING REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130035394-A1 Calixarene-Based Peptide Conformation Mimetics, Methods of Use, and Methods of Making CLSPN, BID, CALU SHBG 470/4885HSPA5 3284/4885HMGB1 2292/4885
US-20120309801-A1 CALIXARENE-BASED PEPTIDE CONFORMATION MIMETICS, METHODS OF USE, AND METHODS OF MAKING CLSPN, BID, CALU SHBG 470/4885HSPA5 3284/4885HMGB1 2292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.