SCHEMBL14214721

SCHEMBL14214721

Bc1ccc(Nc2ncnc(Nc3cc(OC)c(OC)c(OC)c3)n2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 5/20 0.68
EPHB4 P54760 2/20 0.68
KDR P35968 2/20 0.62
AURKB Q96GD4 1/20 0.62
PTK2 Q05397 7/20 0.58
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
FGFR1 P11362 1/20 0.55
FGFR2 P21802 1/20 0.55
FGFR4 P22455 1/20 0.55
FGFR3 P22607 1/20 0.55
EGFR P00533 2/20 0.54
TEK Q02763 1/20 0.54
LCK P06239 1/20 0.52
MAPK14 Q16539 1/20 0.52
JAK2 O60674 1/20 0.49
CDK2 P24941 1/20 0.49
PIK3CA P42336 1/20 0.49
PIK3CB P42338 1/20 0.49
PIK3CG P48736 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6480192 0.81 IGF1R (0.65) IGF1REPHB4KDRAURKBPTK2
SCHEMBL21067672 0.81 EPHB4 (1.00) IGF1REPHB4KDRAURKBPTK2
SCHEMBL14214593 0.80 IGF1R (0.63) IGF1REPHB4KDRAURKBPTK2
SCHEMBL14214584 0.79 IGF1R (0.66) IGF1REPHB4KDRAURKBPTK2
SCHEMBL14214534 0.79 BRD4 (0.60) IGF1REPHB4KDRAURKBPTK2
SCHEMBL4946510 0.78 EPHB4 (0.69) IGF1REPHB4KDRAURKBPTK2
SCHEMBL1927928 0.78 IGF1R (0.61) IGF1REPHB4KDRAURKBPTK2
SCHEMBL13955883 0.78 IGF1R (0.59) IGF1REPHB4KDRAURKBPTK2
SCHEMBL6481952 0.78 EGFR (0.62) IGF1REPHB4KDRAURKBPTK2
SCHEMBL14214750 0.77 IGF1R (0.57) IGF1REPHB4KDRAURKBPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218360-B1 TRIAZINE KINASE INHIBITORS AMGEN INC (US) 2008-05-28 EP disclosed