SCHEMBL14214739

SCHEMBL14214739

COc1cc(Nc2ncnc(-c3cccnc3Nc3cccc(Oc4ccccc4)c3)n2)cc(OC)c1OC

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TEK Q02763 2/20 0.82
KDR P35968 2/20 0.78
FGFR3 P22607 8/20 0.64
FGFR2 P21802 7/20 0.64
IGF1R P08069 4/20 0.53
PTK2 Q05397 1/20 0.48
FGFR1 P11362 1/20 0.48
FGFR4 P22455 1/20 0.48
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48
TUBB3 Q13509 1/20 0.48
TUBB2A Q13885 1/20 0.48
TUBB8 Q3ZCM7 1/20 0.48
TUBA3E Q6PEY2 1/20 0.48
TUBA1A Q71U36 1/20 0.48
TUBA1C Q9BQE3 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14214549 0.90 TEK (0.77) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL6478261 0.88 TEK (1.00) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL6479686 0.84 TEK (0.89) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL6480366 0.84 TEK (0.76) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL6478685 0.84 TEK (0.76) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL6492448 0.83 TEK (0.75) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL14214552 0.83 TEK (0.81) TEKKDRFGFR3FGFR2FGFR1
SCHEMBL6598236 0.82 TEK (0.73) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL14214551 0.81 TEK (0.78) TEKKDRFGFR3FGFR2IGF1R
SCHEMBL14214554 0.81 TEK (0.74) TEKKDRFGFR3FGFR2IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218360-B1 TRIAZINE KINASE INHIBITORS AMGEN INC (US) 2008-05-28 EP disclosed