SCHEMBL14217829

SCHEMBL14217829

N#Cc1ccc2c(c1)C=CCC=N2

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
DRD2 P14416 2/20 0.30
DRD3 P35462 2/20 0.30
PNMT P11086 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24891182 0.74 GAA (0.32)
SCHEMBL1092139 0.69 TRPA1 (0.38) TRPA1CA12CA9NOS3NOS1
SCHEMBL11017385 0.68 TRPA1 (0.44) TRPA1NOS3NOS1NOS2DRD2
SCHEMBL26916671 0.68 TRPA1 (0.35) TRPA1CA12CA9NOS3NOS1
SCHEMBL29740370 0.66 CA1 (0.44) TRPA1CA12CA9DRD2DRD3
SCHEMBL29740368 0.66 CA1 (0.44) TRPA1CA12CA9DRD2DRD3
SCHEMBL148119 0.66 CA1 (0.44) TRPA1CA12CA9DRD2DRD3
SCHEMBL28039609 0.66 PNMT (0.42) TRPA1NOS3NOS1NOS2DRD2
Hydrochloric Acid SCHEMBL20919478 0.65 CA1 (0.43) TRPA1CA12CA9DRD2DRD3
SCHEMBL7038650 0.65 TRPA1 (0.44) TRPA1NOS3NOS1NOS2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060301-A1 7-SUBSTITUTED PURINE DERIVATIVES FOR IMMUNOSUPPRESSION PHARMACOPEIA , LLC (US) 2008-05-22 WO disclosed