SCHEMBL14218592

SCHEMBL14218592

C[N+]1(C)CCN(C2=Cc3ccccc3Oc3ccc(Cl)cc32)CC1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.74
DRD4 P21917 10/20 0.74
TP53 P04637 2/20 0.74
CYP1A2 P05177 2/20 0.74
CYP3A4 P08684 2/20 0.74
CYP2D6 P10635 2/20 0.74
TDP1 Q9NUW8 2/20 0.74
MAPT P10636 1/20 0.74
CYP2C19 P33261 1/20 0.74
HRH4 Q9H3N8 4/20 0.45
HTR3A P46098 3/20 0.45
HRH2 P25021 3/20 0.45
HRH1 P35367 3/20 0.45
ADRB2 P07550 2/20 0.45
CHRM2 P08172 2/20 0.45
CHRM4 P08173 2/20 0.45
HTR1A P08908 2/20 0.45
CHRM5 P08912 2/20 0.45
ADRA2A P08913 2/20 0.45
ADORA3 P0DMS8 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10873714 0.85 DRD2 (1.00) DRD2DRD4TP53CYP1A2CYP3A4
SCHEMBL11932036 0.77 HRH4 (0.74) DRD2DRD4TP53CYP1A2CYP3A4
Fumaric Acid SCHEMBL467100 0.77 DRD4 (0.81) DRD2DRD4TP53CYP1A2CYP3A4
Maleic Acid SCHEMBL467099 0.77 DRD4 (0.81) DRD2DRD4TP53CYP1A2CYP3A4
Fumaric Acid SCHEMBL29699565 0.77 DRD4 (0.81) DRD2DRD4TP53CYP1A2CYP3A4
SCHEMBL11563888 0.77 DRD2 (1.00) DRD2DRD4TP53CYP1A2CYP3A4
SCHEMBL1842504 0.70 DRD2 (0.56) DRD2DRD4TP53CYP1A2CYP3A4
SCHEMBL11577371 0.69 DRD2 (0.67) DRD2DRD4TP53CYP1A2CYP3A4
SCHEMBL11577989 0.68 MAPT (0.56) DRD2DRD4TP53CYP1A2CYP3A4
Metoxepin SCHEMBL2109740 0.68 DRD2 (0.70) DRD2DRD4TP53CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063603-A2 METHODS, COMPOSITIONS, AND KITS FOR TREATING PAIN AND PRURITIS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-05-29 WO disclosed