Pilsicainide

Pilsicainide

SCHEMBL142244

Cc1cccc(C)c1NC(=O)CC12CCCN1CCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 1.00
ATM Q13315 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.48
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
NFKB1 P19838 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPT P10636 3/20 0.44
SCN3A Q9NY46 3/20 0.44
LMNA P02545 3/20 0.44
SCN1A P35498 2/20 0.44
SCN2A Q99250 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pilsicainide SCHEMBL14809244 1.00 KCNH2 (1.00) KCNH2ATML3MBTL1POLBMEN1
Pilsicainide SCHEMBL483632 0.99 KCNH2 (0.97) KCNH2ATML3MBTL1POLBMEN1
Pilsicainide SCHEMBL1650876 0.97 KCNH2 (0.95) KCNH2ATML3MBTL1POLBMEN1
Pilsicainide SCHEMBL14471484 0.97 KCNH2 (0.95) KCNH2ATML3MBTL1POLBMEN1
Pilsicainide SCHEMBL483631 0.97 KCNH2 (0.95) KCNH2ATML3MBTL1POLBMEN1
SCHEMBL15551940 0.85 KCNH2 (0.74) KCNH2L3MBTL1POLBMEN1KMT2A
SCHEMBL10840605 0.80 KCNH2 (0.66) KCNH2POLBKMT2ALMNAALDH1A1
SCHEMBL10371948 0.74 KCNH2 (0.58) KCNH2ATML3MBTL1POLBMEN1
Pyrrocaine SCHEMBL25718 0.72 MEN1 (0.70) KCNH2ATML3MBTL1POLBMEN1
SCHEMBL10372706 0.71 ATM (0.57) KCNH2ATML3MBTL1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 978 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12117453-B2 Predicting patient response to sodium channel blockers WASHINGTON UNIVERSITY (US) 2024-10-15 US claimed
US-20240074968-A1 ORAL PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING PARTICULATE FORMULATION COMPRISING COMPOSITION SUNSHO PHARMACEUTICAL CO LTD (JP) 2024-03-07 US claimed
EP-4279137-A2 ORAL PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING PARTICULATE FORMULATION COMPRISING COMPOSITION Sunsho Pharmaceutical Co., Ltd. (JP) 2023-11-22 EP claimed
EP-3485876-B1 ORAL PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING PARTICULATE FORMULATION COMPRISING COMPOSITION SUNSHO PHARMACEUTICAL CO LTD (JP) 2023-11-22 EP claimed
US-20230201148-A1 USES OF ORNITHINE PHENYLACETATE FOR TREATING HYPERAMMONEMIA MALLINCKRODT LLC 2023-06-29 US claimed
US-11685952-B2 Biomarker for predicting risk of recurrence in patients with paroxysmal atrial fibrillation KOREA UNIVERSITY RESEARCH AND BUSINESS FOUNDATION (KR) 2023-06-27 US claimed
EP-4153162-A1 USES OF ORNITHINE PHENYLACETATE FOR TREATING HYPERAMMONEMIA Ocera Therapeutics, Inc. (US) 2023-03-29 EP claimed
WO-2021236522-A1 USES OF ORNITHINE PHENYLACETATE FOR TREATING HYPERAMMONEMIA OCERA THERAPEUTICS, INC. (US) 2021-11-25 WO claimed
US-20210313015-A1 SPECIFICALLY-SHAPED CRYSTAL OF COMPOUND AND METHOD FOR PRODUCING SAME TOWA PHARMACEUTICAL CO., LTD. (JP) 2021-10-07 US claimed
US-20210228825-A1 METHODS FOR DIAGNOSING BRUGADA SYNDROME USING AN AEROSOL DEERFIELD MANAGEMENT COMPANY, L.P. (SERIES C), AS COLLATERAL AGENT 2021-07-29 US claimed
WO-2004056181-A1 ORGAN PRECONDITIONING, ARREST, PROTECTION, PRESERVATION AND RECOVERY (2) GLOBAL CARDIAC SOLUTIONS PTY LTD (AU) 2004-07-08 WO claimed
WO-2004056180-A1 ORGAN PRECONDITIONING, ARREST, PROTECTION, PRESERVATION AND RECOVERY (1) GLOBAL CARDIAC SOLUTIONS PTY LTD (AU) 2004-07-08 WO claimed
US-20040087513-A1 New drug combinations based on sodium channel blockers and magnesium salts BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-06 US claimed
WO-2004019909-A2 BUCCAL, POLAR AND NON-POLAR SPRAY OR CAPSULE CONTAINING CARDIOVASCULAR OR RENAL DRUGS NOVADEL PHARMA INC. (US) 2004-03-11 WO claimed
WO-2004004723-A1 NOVEL MEDICAMENT COMBINATIONS BASED ON SODIUM CHANNEL BLOCKERS AND MAGNESIUM SALTS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-01-15 WO claimed
US-20030235576-A1 New drug combinations for the treatment of ischaemic conditions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-12-25 US claimed
WO-2003105844-A1 MEDICAMENT COMBINATIONS OF SODIUM CHANNEL BLOCKERS AND FIBRINOLYTICS FOR TREATING ISCHAEMIC CONDITIONS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-12-24 WO claimed
US-20030077229-A1 Buccal, polar and non-polar spray or capsule containing cardiovascular or renal drugs NOVADEL PHARMA INC. 2003-04-24 US claimed
EP-0089061-B1 8-SUBSTITUTED PYRROLIZIDINE DERIVATIVES AND USE THEREOF SUNTORY KABUSHIKI KAISHA (JP) 1987-12-16 EP claimed
US-4564624-A 8-(Substituted N-phenylcarboxamidomethyl) pyrrolizidines and use thereof as antiarrhythmics SUNTORY LTD. (JP) 1986-01-14 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087513-A1 New drug combinations based on sodium channel blockers and magnesium salts CACNA1B, CACNA1C, CACNA1D KCNH2 53/4885ATM 4593/4885L3MBTL1 4789/4885
US-20210313015-A1 SPECIFICALLY-SHAPED CRYSTAL OF COMPOUND AND METHOD FOR PRODUCING SAME NOTUM, SOAT1, GYS2 KCNH2 2037/4885ATM 2994/4885L3MBTL1 4856/4885
US-20030235576-A1 New drug combinations for the treatment of ischaemic conditions SCN1B, CACNA1B, TNNI3 KCNH2 34/4885ATM 4501/4885L3MBTL1 4643/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.