SCHEMBL14224450

SCHEMBL14224450

CCN(CC)CCNc1cccc(Nc2nccc(-c3cnc(-c4cccnc4)[nH]3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 18/20 0.48
BCR P11274 15/20 0.48
CDK4 P11802 2/20 0.47
CDK2 P24941 2/20 0.47
GSK3B P49841 2/20 0.47
PRKCA P17252 9/20 0.47
SRC P12931 9/20 0.47
PRKCD Q05655 7/20 0.47
PDGFRB P09619 6/20 0.47
PDGFRA P16234 6/20 0.47
EGFR P00533 3/20 0.46
PRKACA P17612 1/20 0.46
PRKACG P22612 1/20 0.46
PRKACB P22694 1/20 0.46
ABL2 P42684 1/20 0.44
PRKD3 O94806 1/20 0.44
PRKCG P05129 1/20 0.44
PRKCB P05771 1/20 0.44
PRKCH P24723 1/20 0.44
PRKCI P41743 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14224139 0.86 ABL1 (0.63) ABL1BCRPRKCASRCPRKCD
SCHEMBL14224448 0.78 KIT (0.54) ABL1BCRGSK3BPRKCASRC
SCHEMBL14224137 0.78 ABL1 (0.66) ABL1BCRPRKCASRCPRKCD
SCHEMBL14196033 0.78 ABL1 (0.54) ABL1BCRPRKCASRCPRKCD
SCHEMBL13924611 0.76 SYK (0.63) CDK4CDK2GSK3BSRC
SCHEMBL14196037 0.75 ABL1 (0.64) ABL1BCRPRKCASRCPRKCD
SCHEMBL14224452 0.75 ABL1 (0.50) ABL1BCRPRKCASRCPRKCD
SCHEMBL14195964 0.75 ABL1 (0.56) ABL1BCRPRKCASRCPRKCD
SCHEMBL14224269 0.75 ABL1 (0.51) ABL1BCRCDK4CDK2GSK3B
SCHEMBL14196032 0.74 ABL1 (0.56) ABL1BCRPRKCASRCPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361665-B2 Inhibitors of c-Jun N-terminal kinases (JNK) and other protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-04-22 US disclosed