SCHEMBL14224673

SCHEMBL14224673

Cn1cc(NC(=O)c2cc3ccccc3cn2)cc1C(=O)Nc1cc(-c2nc3cc(OCCN4CCOCC4)ccc3[nH]2)n(C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.45
PDGFRA P16234 1/20 0.45
KDR P35968 2/20 0.41
FGFR1 P11362 2/20 0.41
ACHE P22303 2/20 0.41
RUNX1 Q01196 2/20 0.40
CFTR P13569 1/20 0.40
LTA4H P09960 1/20 0.40
GRM4 Q14833 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NR3C1 P04150 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
AURKB Q96GD4 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14224528 0.89 KDM4E (0.43) ACHEKDM4ENPC1ALDH1A1TP53
SCHEMBL14427363 0.82 MAPT (0.39) PDGFRBPDGFRANPC1RAB9AABCB1
SCHEMBL14426980 0.82 MAPT (0.39) PDGFRBPDGFRARAB9AABCB1ABCG2
SCHEMBL14224537 0.81 MAPT (0.39) PDGFRBPDGFRANPC1RAB9AABCB1
SCHEMBL14224534 0.79 MAPT (0.40) PDGFRBPDGFRAKDM4ENPC1ALDH1A1
SCHEMBL14426984 0.77 MAPT (0.41) PDGFRBPDGFRANPC1TP53RAB9A
SCHEMBL14224680 0.75 ACHE (0.54) PDGFRBPDGFRAKDRFGFR1ACHE
SCHEMBL14224672 0.73 ACHE (0.50) PDGFRBPDGFRAKDRFGFR1ACHE
SCHEMBL14224524 0.72 MAPT (0.37) ACHEKDM4ENPC1TP53RAB9A
SCHEMBL3382470 0.69 KDR (0.60) PDGFRBPDGFRAKDRFGFR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090816-A1 ANTI-INFECTIVE BIARYL COMPOUNDS GENESOFT PHARMACEUTICALS, INC. (US) 2008-04-17 US disclosed
US-7265129-B2 Anti-infective biaryl compounds GENESOFT PHARMACEUTICALS, INC. (US) 2007-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080090816-A1 ANTI-INFECTIVE BIARYL COMPOUNDS QTRT1, Q6ZSR9, QTRT2 PDGFRB 3401/4885PDGFRA 3599/4885KDR 3146/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.