SCHEMBL14229192

SCHEMBL14229192

CCCCN(C(C)C)S(=O)(=O)CCOCC(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PLA2G2C Q5R387 1/20 0.35
CES1 P23141 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14228927 0.89 CES1 (0.33) CES1
SCHEMBL14229459 0.83 PLA2G2C (0.37) PLA2G2CCES1CYP2C9TSHRCYP2C19
SCHEMBL14200405 0.82
SCHEMBL14230127 0.82 PLA2G2C (0.35) PLA2G2CCES1CYP2C9TSHRCYP2C19
SCHEMBL14229464 0.81 PLA2G2C (0.35) PLA2G2CCES1CYP2C9TSHRCYP2C19
SCHEMBL14229190 0.80 CES1 (0.33) CES1
SCHEMBL14229150 0.77 PLA2G2C (0.33) PLA2G2CCES1CYP2C9TSHRCYP2C19
SCHEMBL14200391 0.76 PLA2G2C (0.33) PLA2G2CCES1
SCHEMBL14229116 0.75 TP53 (0.35) HSD17B10
SCHEMBL14229376 0.73 CA2 (0.41) CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed