SCHEMBL14229247

SCHEMBL14229247

CCCCN(Cc1cccc(C)c1)C(=O)CCC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.51
GRIN3B O60391 1/20 0.51
GRIN1 Q05586 1/20 0.51
GRIN2A Q12879 1/20 0.51
GRIN2B Q13224 1/20 0.51
GRIN2C Q14957 1/20 0.51
GRIN3A Q8TCU5 1/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC2 Q92769 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
LTB4R2 Q9NPC1 2/20 0.47
CNR2 P34972 1/20 0.46
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
PAX8 Q06710 2/20 0.46
TP53 P04637 1/20 0.46
GPX4 P36969 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14228983 0.92 GRIN2D (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14200916 0.85 GRIN2D (0.48) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14229453 0.84 LTB4R2 (0.62) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229062 0.83 BCHE (0.54) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14229430 0.82 HDAC6 (0.54) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9327545 0.78 CNR2 (0.61) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229063 0.78 HDAC1 (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14229228 0.78 TSHR (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14229226 0.77 CTSB (0.40) LTB4R2ALDH1A1NPC1RAB9APAX8
SCHEMBL14229121 0.77 TP53 (0.69) LTB4R2ALDH1A1NPC1RAB9APAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed