SCHEMBL14229063

SCHEMBL14229063

CCCCN(Cc1ccc(F)c(F)c1)C(=O)CCC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC3 O15379 1/20 0.53
HDAC2 Q92769 1/20 0.53
NCOR2 Q9Y618 1/20 0.53
RIPK1 Q13546 1/20 0.46
LTB4R2 Q9NPC1 3/20 0.45
CNR2 P34972 2/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MITF O75030 1/20 0.42
HTT P42858 1/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
LPAR1 Q92633 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229280 0.92 RIPK1 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200903 0.85 RIPK1 (0.49) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229430 0.82 HDAC6 (0.54) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229228 0.81 TSHR (0.53) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229225 0.78 HDAC3 (0.51) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229453 0.78 LTB4R2 (0.62) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229247 0.78 GRIN2D (0.51) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229234 0.77 RIPK1 (0.43) RIPK1LTB4R2ALDH1A1KDM4EMITF
SCHEMBL14200852 0.77 RIPK1 (0.51) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14228980 0.76 RIPK1 (0.42) RIPK1LTB4R2ALDH1A1KDM4EMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed