SCHEMBL14237115

SCHEMBL14237115

COc1ccc2c(c1)CCN(C(C1CCCNC1)S(=O)(=O)c1ccccc1Cl)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.39
DRD1 P21728 2/20 0.39
DRD5 P21918 1/20 0.39
HTR2C P28335 3/20 0.38
HTR2B P41595 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
USP30 Q70CQ3 1/20 0.37
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALK Q9UM73 1/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1628038 0.99 HTR6 (0.38) HTR6DRD1DRD5HTR2CHTR2B
SCHEMBL14237116 0.91 HTR6 (0.38) HTR6DRD1DRD5HTR2CHTR2B
Hydrochloric Acid SCHEMBL1628011 0.90 HTR6 (0.37) HTR6HTR2CHTR2BUSP30LMNA
Hydrochloric Acid SCHEMBL1627613 0.90 ALK (0.41) ALK
SCHEMBL14236970 0.89 DRD1 (0.41) HTR6DRD1DRD5HTR2CALDH1A1
Hydrochloric Acid SCHEMBL1627851 0.89 DRD1 (0.40) HTR6DRD1DRD5HTR2CALDH1A1
SCHEMBL14237049 0.88 HTR6 (0.39) HTR6HTR2CALDH1A1HPGDMAPT
SCHEMBL14237162 0.88 HTR2C (0.37) HTR6DRD1DRD5HTR2CHTR2B
Hydrochloric Acid SCHEMBL1625893 0.88 NPY5R (0.42) HTR6
SCHEMBL14237023 0.88 AKR1C3 (0.41) HTR6DRD1DRD5HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831195-B1 5-HT7 RECEPTOR ANTAGONISTS ESTEVE LABOR DR (ES) 2012-12-19 EP claimed