Bicarbonate

Bicarbonate

SCHEMBL14237153

Cc1cccc(C2(C)C=CCC(C)C2)c1.O=C(O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A known ✓ P49840 1/20 0.38
GSK3B known ✓ P49841 1/20 0.38
CCR2 P41597 11/20 0.57
HCAR2 Q8TDS4 1/20 0.41
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
SLC6A2 P23975 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CHRND Q07001 1/20 0.39
HDAC4 P56524 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL14237131 0.86 CCR2 (0.54) CCR2
Bicarbonate SCHEMBL14237102 0.85 CCR2 (0.58) CCR2HCAR2CHRNA1CHRNB1CHRNB2
Bicarbonate SCHEMBL14237231 0.85 CCR2 (0.58) CCR2CHRNA1CHRNGCHRNB1CHRNB2
Bicarbonate SCHEMBL14237083 0.83 CCR2 (0.54) CCR2CHRNA1CHRNGCHRNB1CHRNB2
Bicarbonate SCHEMBL14237258 0.82 CCR2 (0.56) CCR2HPGD
Bicarbonate SCHEMBL14237114 0.82 CCR2 (0.61) CCR2HCAR2KMT2AOPRM1EPHX2
SCHEMBL28842376 0.79 CCR2 (0.45) CCR2
Bicarbonate SCHEMBL14237079 0.79 CCR2 (0.47) CCR2MEN1KMT2A
Bicarbonate SCHEMBL14237166 0.79 CCR2 (0.46) CCR2
Bicarbonate SCHEMBL14237132 0.77 CCR2 (0.44) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318352-B1 CYCLOHEXENYL COMPOUNDS AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-12-19 EP claimed