Bicarbonate

Bicarbonate

SCHEMBL14237231

CC1CC=CC(C)(c2cccc(-c3ccccc3)c2)C1.O=C(O)O

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 14/20 0.58
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
CHRND Q07001 1/20 0.36
KMO O15229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL14237153 0.85 CCR2 (0.57) CCR2SLC6A2SLC6A3CHRNA1CHRNG
Bicarbonate SCHEMBL14237102 0.84 CCR2 (0.58) CCR2SLC6A2SLC6A4SLC6A3CHRNA1
SCHEMBL28842376 0.81 CCR2 (0.45) CCR2
Bicarbonate SCHEMBL14237114 0.81 CCR2 (0.61) CCR2
Bicarbonate SCHEMBL14237258 0.78 CCR2 (0.56) CCR2
Bicarbonate SCHEMBL14237131 0.76 CCR2 (0.54) CCR2
Bicarbonate SCHEMBL14237079 0.75 CCR2 (0.47) CCR2KMO
Bicarbonate SCHEMBL14237166 0.75 CCR2 (0.46) CCR2
Bicarbonate SCHEMBL14237273 0.75 CCR2 (0.55) CCR2
SCHEMBL1780947 0.74 CCR2 (1.00) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318352-B1 CYCLOHEXENYL COMPOUNDS AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-12-19 EP claimed