Bicarbonate

Bicarbonate

SCHEMBL14237192

C[C@@H]1CC=C[C@](C)(c2ccc(Cl)c(C(F)(F)F)c2)C1.O=C(O)O

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 11/20 0.62
OPRM1 P35372 3/20 0.37
GRIN2B Q13224 2/20 0.37
OPRD1 P41143 2/20 0.37
OPRL1 P41146 2/20 0.37
NOTUM Q6P988 3/20 0.37
KDR P35968 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL14237107 1.00 CCR2 (0.62) CCR2OPRM1GRIN2BOPRD1OPRL1
Bicarbonate SCHEMBL14237203 0.85 CCR2 (0.63) CCR2OPRM1GRIN2BOPRD1OPRL1
Bicarbonate SCHEMBL14237150 0.85 CCR2 (0.63) CCR2OPRM1GRIN2BOPRD1OPRL1
Bicarbonate SCHEMBL14237270 0.81 CCR2 (0.48) CCR2OPRM1GRIN2BOPRD1OPRL1
Bicarbonate SCHEMBL14237136 0.81 CCR2 (0.66) CCR2OPRM1GRIN2BOPRD1OPRL1
Bicarbonate SCHEMBL14237079 0.81 CCR2 (0.47) CCR2
Bicarbonate SCHEMBL14237114 0.79 CCR2 (0.61) CCR2OPRM1GRIN2BOPRL1
Bicarbonate SCHEMBL14237147 0.78 CCR2 (0.57) CCR2
SCHEMBL14237157 0.78 CCR2 (0.61) CCR2
SCHEMBL1781364 0.77 CCR2 (1.00) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318352-B1 CYCLOHEXENYL COMPOUNDS AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-12-19 EP claimed