SCHEMBL14237352

SCHEMBL14237352

CCNC(=O)c1nc(-c2cccc(C(=O)O)c2C)cnc1N

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.57
LDHB P07195 1/20 0.57
ATR Q13535 18/20 0.52
PRKDC P78527 6/20 0.52
ACVR1 Q04771 1/20 0.52
ATM Q13315 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14237367 0.83 LDHA (0.60) LDHALDHBATRPRKDCATM
SCHEMBL14237502 0.83 ACVR2A (0.55) LDHALDHBATRPRKDCACVR1
SCHEMBL3460516 0.77 ATR (0.70) LDHALDHBATRPRKDCACVR1
SCHEMBL3462214 0.74 ACVR1 (0.61) ATRPRKDCACVR1ATM
SCHEMBL3460485 0.72 ACVR1 (0.61) ATRPRKDCACVR1ATM
SCHEMBL3460037 0.71 ACVR1 (0.57) ATRPRKDCACVR1
SCHEMBL3461134 0.71 ACVR1 (0.63) ATRPRKDCACVR1ATM
SCHEMBL3460825 0.70 ATR (0.58) LDHALDHBATRPRKDCACVR1
SCHEMBL17434318 0.70 ATR (0.56) ATRPRKDCACVR1
SCHEMBL11909154 0.69 ATR (0.72) LDHALDHBATRPRKDCATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501514-B1 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2012-12-19 EP claimed