SCHEMBL14237367

SCHEMBL14237367

Cc1c(C(=O)O)cccc1-c1cnc(N)c(C(N)=O)n1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.60
LDHB P07195 1/20 0.60
ATR Q13535 18/20 0.49
PRKDC P78527 6/20 0.49
ATM Q13315 3/20 0.43
MYC P01106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14237352 0.83 LDHA (0.57) LDHALDHBATRPRKDCATM
SCHEMBL14237502 0.82 ACVR2A (0.55) LDHALDHBATRPRKDC
SCHEMBL3461548 0.80 ATR (0.68) LDHALDHBATRPRKDCATM
SCHEMBL3459735 0.76 ATR (0.50) ATRPRKDCATM
SCHEMBL3461447 0.74 ATR (0.68) ATRPRKDCATM
SCHEMBL11909154 0.74 ATR (0.72) LDHALDHBATRPRKDCATM
SCHEMBL3460267 0.74 ATR (0.70) LDHALDHBATRPRKDCATM
SCHEMBL24248259 0.73 ATR (0.67) ATRPRKDCATM
SCHEMBL3460629 0.72 ATR (0.68) ATRPRKDCATM
SCHEMBL3460235 0.72 ATR (0.70) LDHALDHBATRPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501514-B1 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2012-12-19 EP claimed