SCHEMBL14237643

SCHEMBL14237643

COc1cc2cc(OC(=O)NCC(C)(C)N(C)C)c3c4cc5c(cc4ncc3c2cc1OC)OCO5

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 8/20 0.37
NQO1 P15559 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HTT P42858 2/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SLC6A5 Q9Y345 1/20 0.35
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
PDE10A Q9Y233 3/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PDE5A O76074 1/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14237587 0.92 TDP1 (0.36) TDP1NQO1ALDH1A1HTTLMNA
SCHEMBL14237632 0.90 TDP1 (0.37) TDP1NQO1ALDH1A1HTTLMNA
SCHEMBL2129981 0.88 SLC6A5 (0.38) TDP1NQO1ALDH1A1HTTLMNA
SCHEMBL2130106 0.82 ALDH1A1 (0.36) TDP1ALDH1A1HTTLMNANPSR1
SCHEMBL1726191 0.80 TDP1 (0.37) TDP1ALDH1A1HTTLMNANPSR1
SCHEMBL1724918 0.79 SLC6A5 (0.41) TDP1ALDH1A1HTTLMNANPSR1
SCHEMBL2601747 0.76 RAD52 (0.42) TDP1ALDH1A1HTTLMNANPSR1
SCHEMBL2601755 0.75 ALDH1A1 (0.45) NQO1ALDH1A1HTTLMNANPSR1
SCHEMBL2601754 0.75 ALDH1A1 (0.45) TDP1NQO1ALDH1A1HTTLMNA
SCHEMBL2601756 0.74 ALDH1A1 (0.44) TDP1NQO1ALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403856-B1 METHYLENEDIOXYBENZO [I]PHENANTHRIDINE DERIVATIVES USED TO TREAT CANCER UNIV RUTGERS (US) 2012-12-19 EP claimed