SCHEMBL14239113

SCHEMBL14239113

CC1CCn2c(nc3cc(-c4ccccn4)cnc3c2=O)C1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.39
MAPT P10636 3/20 0.38
TP53 P04637 3/20 0.38
CNR2 P34972 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
TGFBR1 P36897 1/20 0.34
METAP2 P50579 1/20 0.34
TNKS O95271 1/20 0.34
DHFR P00374 1/20 0.34
USP30 Q70CQ3 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239109 0.94 CNR2 (0.37) LMNAMAPTTP53CNR2HRH3
SCHEMBL6922373 0.91 MAPT (0.37) LMNAMAPTTP53CNR2HRH3
SCHEMBL6923220 0.89 MAPT (0.36) MAPTCNR2HRH3GSK3BDYRK1A
SCHEMBL14240248 0.87 SMO (0.36) CNR2HRH3GSK3BDYRK1ATGFBR1
SCHEMBL6920417 0.86 NPC1 (0.41) LMNAMAPTTP53GSK3BDYRK1A
SCHEMBL14239310 0.85 METAP2 (0.38) CNR2HRH3GSK3BDYRK1ATGFBR1
SCHEMBL14239107 0.83 USP30 (0.35) LMNAMAPTTP53CNR2HRH3
SCHEMBL14238856 0.83 METAP2 (0.34) CNR2HRH3GSK3BDYRK1ATGFBR1
SCHEMBL14239108 0.82 SMO (0.39) LMNATP53CNR2HRH3GSK3B
SCHEMBL14239044 0.82 TGFBR1 (0.36) LMNATP53CNR2HRH3GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed