SCHEMBL14239372

SCHEMBL14239372

O=c1c2ccc(-c3ccccn3)cc2nc2n1CC1(C2)CC1(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
CYP3A4 P08684 1/20 0.36
NSD2 O96028 1/20 0.36
METAP2 P50579 2/20 0.35
TGFBR1 P36897 1/20 0.34
DHODH Q02127 1/20 0.34
PRMT5 O14744 2/20 0.34
WDR77 Q9BQA1 1/20 0.34
PIK3CD O00329 4/20 0.33
PIK3CA P42336 4/20 0.33
PIK3CG P48736 4/20 0.33
PI4KA P42356 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
PIK3CB P42338 2/20 0.33
BACE1 P56817 2/20 0.32
CTSD P07339 1/20 0.32
ABL1 P00519 1/20 0.32
RET P07949 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239321 0.90 NPC1 (0.39) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14239346 0.88 NPC1 (0.42) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL12059073 0.84 NPC1 (0.40) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL6922046 0.83 NPC1 (0.42) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL6922549 0.82 NPC1 (0.36) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14238863 0.80 NPC1 (0.40) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14239067 0.80 METAP2 (0.40) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14239105 0.80 POLB (0.41) NPC1RAB9ATDP1NSD2
SCHEMBL14240301 0.79 NPC1 (0.42) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL12059030 0.79 NPC1 (0.42) NPC1RAB9ATDP1CYP3A4NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed